TargetMol

hCAIX-IN-5

Product Code:
 
TAR-T60745
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T60745-1mg1mg£227.00
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TAR-T60745-5mg5mg£458.00
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Quantity:
TAR-T60745-10mg10mg£626.00
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TAR-T60745-25mg25mg£938.00
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Quantity:
TAR-T60745-50mg50mg£1,267.00
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Quantity:
TAR-T60745-100mg100mg£1,653.00
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Quantity:
TAR-T60745-500mg500mg£3,227.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.
CAS:
2451479-57-3
Molecular Weight:
309.29
Pathway:
Metabolism
Purity:
0.98
SMILES:
N(C(/C=C/C1=CC=C(F)C=C1)=O)C=2C=C3C(=CC2)OC(=O)C=C3
Target:
Carbonic Anhydrase

References

Swain B, et al. New coumarin/sulfocoumarin linked phenylacrylamides as selective transmembrane carbonic anhydrase inhibitors: Synthesis and in-vitro biological evaluation. Bioorg Med Chem. 2020 Aug 1;28(15):115586.