TargetMol

MMP2-IN-3

Product Code:
 
TAR-T61271
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T61271-1mg1mg£189.00
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Quantity:
TAR-T61271-5mg5mg£343.00
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TAR-T61271-1mL1 mL * 10 mM (in DMSO)£358.00
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TAR-T61271-10mg10mg£483.00
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TAR-T61271-25mg25mg£743.00
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Quantity:
TAR-T61271-50mg50mg£1,002.00
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Quantity:
TAR-T61271-100mg100mg£1,324.00
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Quantity:
TAR-T61271-500mg500mg£2,577.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 uM). MMP2-IN-3 inhibits MMP-9 and MMP-8 with IC50s of 26.6 and 32 uM, respectively.
CAS:
897799-81-4
Molecular Weight:
355.43
Pathway:
Proteases/Proteasome
Purity:
0.9913
SMILES:
O=C(NC1=CC=CC(=C1)C2=NC3=CC(=CC=C3N2)C)CCC=4C=CC=CC4
Target:
MMP

References

Laghezza A, et al. Virtual screening identification and chemical optimization of substituted 2-arylbenzimidazoles as new non-zinc-binding MMP-2 inhibitors. Bioorg Med Chem. 2020 ; 28(3):115257.