TargetMol

AGI-41998 tautomers

Product Code:
 
TAR-T64377
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T64377-1mg1mg£227.00
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TAR-T64377-5mg5mg£430.00
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TAR-T64377-1mL1 mL * 10 mM (in DMSO)£507.00
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TAR-T64377-10mg10mg£600.00
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TAR-T64377-25mg25mg£863.00
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TAR-T64377-50mg50mg£1,179.00
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TAR-T64377-100mg100mg£1,589.00
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TAR-T64377-500mg500mg£3,115.00
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Further Information

Bioactivity:
AGI-41998 tautomers is a tautomerism of pyrido[4,3-d]pyrimidin-7(6H)-one, 8-(4-bromophenyl)-6-(4-methoxyphenyl)-2-[(2,2,2-trifluoroethyl)amino]-. pyrido[4,3-d]pyrimidin-7(6H)-one, 8-(4-bromophenyl)-6-(4-methoxyphenyl)-2-[(2,2,2-trifluoroethyl)amino]- is a S-adenosylmethionine synthase isoform type-2 inhibitor, IC50= 0.022uM.
CAS:
T64377
Molecular Weight:
505.29
Purity:
0.9958
SMILES:
O=C1C(C2=CC=C(Br)C=C2)=C(C(C=N3)=CN1C4=CC=C(OC)C=C4)NC3=NCC(F)(F)F

References

Li M, et al. Leveraging Structure-Based Drug Design to Identify Next-Generation MAT2A Inhibitors, Including Brain-Penetrant and Peripherally Efficacious Leads. J Med Chem. 2022 Mar 24;65(6):4600-4615.