TargetMol

GW 833972A

Product Code:
 
TAR-T64394
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T64394-1mg1mg£352.00
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TAR-T64394-5mg5mg£736.00
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TAR-T64394-1mL1 mL * 10 mM (in DMSO)£868.00
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TAR-T64394-10mg10mg£978.00
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TAR-T64394-25mg25mg£1,348.00
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TAR-T64394-50mg50mg£1,661.00
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Quantity:
TAR-T64394-100mg100mg£2,079.00
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Quantity:
TAR-T64394-500mg500mg£4,006.00
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  • Further Information
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Further Information

Bioactivity:
GW 833972A is a selective CB2 receptor agonist.GW 833972A has an inhibitory effect on induced neural depolarization and on citric acid-induced cough in an animal model.
CAS:
1092502-33-4
Molecular Weight:
727.93
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
O(C)C1=C2C=[N+]3C(C=4C(=CC5=C(C4)OCO5)CC3)=CC2=CC=C1OC.C[C@@]12[C@]([C@]3([C@@]([C@]4(C)[C@](C[C@@H]3O)(C[C@H](O)CC4)[H])(CC1)[H])[H])(CC[C@@]2([C@@H](CCC([O-])=O)C)[H])[H]
Target:
Cannabinoid Receptor

References

Belvisi MG, et al. Inhibitory activity of the novel CB2 receptor agonist, GW833972A, on guinea-pig and human sensory nerve function in the airways. Br J Pharmacol. 2008;155(4):547-557. Takheaw N, et al. Cannabinoid Receptor 1 Agonist ACEA and Cannabinoid Receptor 2 Agonist GW833972A Attenuates Cell-Mediated Immunity by Different Biological Mechanisms. Cells. 2023;12(6):848. S?nchez-Zavaleta R, et al. Presynaptic cannabinoid CB2 receptors modulate [3 H]-Glutamate release at subthalamo-nigral terminals of the rat. Synapse. 2018;72(11):e22061.