TargetMol

CB2R/FAAH?modulator-2

Product Code:
 
TAR-T67745
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T67745-1mg1mg£95.00
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TAR-T67745-5mg5mg£128.00
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TAR-T67745-1mL1 mL * 10 mM (in DMSO)£140.00
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TAR-T67745-10mg10mg£168.00
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TAR-T67745-25mg25mg£230.00
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TAR-T67745-50mg50mg£309.00
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Quantity:
TAR-T67745-100mg100mg£434.00
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Further Information

Bioactivity:
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-2 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 10.8 and 152.9 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 6.2 uM. CB2R/FAAH modulator-2 has studies research value related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.
CAS:
2876918-68-0
Molecular Weight:
367.52
Pathway:
Neuroscience|GPCR/G Protein|Metabolism
Purity:
0.9952
SMILES:
O=C(NC12CC3CC(CC(C3)C1)C2)C=4C=CC=CC4OCC5CCCCC5
Target:
Cannabinoid Receptor|FAAH

References

Francesca Intranuovo, et al. Development of N-(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. J Med Chem. 2023 Jan 12;66(1):235-250.