TargetMol

Pirodomast

Product Code:
 
TAR-T67959
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T67959-1mg1mg£201.00
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TAR-T67959-5mg5mg£384.00
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TAR-T67959-10mg10mg£544.00
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TAR-T67959-25mg25mg£828.00
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TAR-T67959-50mg50mg£1,099.00
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Quantity:
TAR-T67959-100mg100mg£1,460.00
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Quantity:
TAR-T67959-500mg500mg£2,850.00
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This product comes from: United States.
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Further Information

Bioactivity:
Pirodomast is a thromboxane A (TXA2) synthase inhibitor. Pirodomast inhibits leukotriene (LT) D4, C4, E4 formation and thromboxane B2 (TXB2) activity, but is weakly or ineffectively antagonistic to guinea pig bronchospasm induced by histamine, methacholine, serotonin, LTC4, or platelet-activating factor. Pirodomast is a potential antiallergic compound. Pirodomast had only weak relaxant activity on guinea pig trachea in vitro. Pirodomast is a potential antiallergic compound that inhibits the protein hydrolyzing activity of trypsin in vitro, prevents antigen-induced immediate and late asthmatic responses in allergic sheep in vivo, and inhibits antigen-induced airway hyperresponsiveness to histamine and carbachol in allergic sheep.
CAS:
108310-20-9
Formula:
C18H17N3O2
Molecular Weight:
307.35
Pathway:
Proteases/Proteasome
Purity:
0.9934
SMILES:
O=C1C2=CC=CN=C2N(C=3C=CC=CC3)C(=O)C1N4CCCC4
Target:
Thrombin|Serine Protease

References

Mizushima Y, et al. Clinical potential of anti-thromboxane A2 agents in bronchial asthma. BioDrugs. 1997; 7(2): 91-98.