TargetMol

ERRγ Inverse Agonist 1

Product Code:
 
TAR-T11231
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T11231-5mg5mg£850.00
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TAR-T11231-50mg50mg£1,661.00
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Quantity:
TAR-T11231-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
CAS:
2316832-86-5
Formula:
C30H38Cl2N2O2
Molecular Weight:
529.54
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
OC1=CC=CC(/C(C2=CC=C(N3CCN(C(C)C)CC3)C=C2)=C(C4=CC=CC=C4)\CCCO)=C1.[H]Cl.[H]Cl
Target:
Estrogen/progestogen Receptor

References

Kim J, et al. Discovery of Potent, Selective, and Orally Bioavailable Estrogen-Related Receptor-? Inverse Agonists To Restore the Sodium Iodide Symporter Function in Anaplastic Thyroid Cancer. J Med Chem. 2019 Feb 28;62(4):1837-1858.