TargetMol

8-CPT-2Me-cAMP, sodium salt

Product Code:
 
TAR-T22014
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T22014-5mg5mg£430.00
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TAR-T22014-50mg50mg£986.00
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Quantity:
TAR-T22014-100mg100mg£1,532.00
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Further Information

Bioactivity:
8-CPT-2Me-cAMP sodium is a sodium salt compound that selectively activates exchange proteins activated by cAMP (Epac). These Epac proteins are cAMP-sensitive guanine nucleotide exchange factors (GEFs) responsible for activating small GTPases Rap1 and Rap2. 8-CPT-2Me-cAMP sodium specifically activates Epac1 with an EC50 value of 2.2 uM, while showing no activation of PKA with an EC50 value greater than 10 uM [1]. Additionally, 8-CPT-2Me-cAMP sodium stimulates the Epac-mediated release of calcium ions (Ca2+) in vitro in pancreatic β-cells [2].
CAS:
634207-53-7
Molecular Weight:
507.82
Purity:
0.98
SMILES:
[Na+].CO[C@@H]1[C@@H]2OP([O-])(=O)OC[C@H]2O[C@H]1n1c(Sc2ccc(Cl)cc2)nc2c(N)ncnc12