TargetMol

NAAA-IN-3

Product Code:
 
TAR-T60432
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T60432-5mg5mg£850.00
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Quantity:
TAR-T60432-50mg50mg£1,661.00
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Quantity:
TAR-T60432-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
NAAA-IN-3 (Compound 17a) is a potent and selective NAAA inhibitor with an IC50 of 50 nM. NAAA is a cysteine amidase which preferentially hydrolyzes the endogenous biolipids palmitoylethanolamide (PEA) and oleoylethanolamide (OEA). PEA is an endogenous agonist of the nuclear peroxisome proliferator-activated receptor-α (PPAR-α), which is a key regulator of inflammation and pain. The potential role of NAAA-IN-3 is as a therapeutic agent for the treatment of inflammation and pain.
CAS:
1831115-59-3
Molecular Weight:
264.328
Purity:
0.98
SMILES:
N#CN1CC(C1)OCc1ccc(cc1)-c1ccccc1