TargetMol

(R)-STU104

Product Code:
 
TAR-T60657
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T60657-5mg5mg£850.00
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Quantity:
TAR-T60657-50mg50mg£1,661.00
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Quantity:
TAR-T60657-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
(R)-STU104 is a potent and orally active TAK1-MKK3 interaction inhibitor that can be used in ulcerative colitis research. (R)-STU104 has IC50s of 0.58 uM and 4.0 uM for the phosphorylation of TNF-α and MKK3. (R)-STU104 binds with MKK3 and disrupts the TAK1 phosphorylating MKK3 to suppress the TAK1/MKK3/p38/MnK1/MK2/elF4E signal pathways [1].
CAS:
2767124-77-4
Molecular Weight:
298.338
Purity:
0.98
SMILES:
COc1ccc(cc1)[C@H]1CC(=O)c2cc(OC)cc(OC)c12