TargetMol

Protein kinase D inhibitor 1

Product Code:
 
TAR-T61163
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61163-5mg5mg£850.00
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Quantity:
TAR-T61163-50mg50mg£1,661.00
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Quantity:
TAR-T61163-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Protein kinase D inhibitor 1 (compound 17m) is a potent pan-PKD inhibitor. It exhibits inhibitory activity in the low nanomolar range, with IC50 values ranging between 17 and 35 nM. By inhibiting protein kinase D, this compound effectively suppresses cortactin phosphorylation, which is known to be PKD-dependent [1].
CAS:
2489320-03-6
Molecular Weight:
347.426
Purity:
0.98
SMILES:
Nc1ncnc2n(CC3CCNCC3)nc(-c3c[nH]c4ccccc34)c12