TargetMol

Irdabisant hydrochloride

Product Code:
 
TAR-T61197
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61197-5mg5mg£850.00
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TAR-T61197-50mg50mg£1,661.00
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Quantity:
TAR-T61197-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Irdabisant (CEP-26401) hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist with K i values of 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively. Irdabisant hydrochloride has relatively low inhibitory activity against hERG current with an IC 50 of 13.8 uM. Irdabisant hydrochloride has cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant hydrochloride can be used to research schizophrenia or cognitive impairment [1] [2].
CAS:
1005398-61-7
Formula:
C18H24ClN3O2
Molecular Weight:
349.86
Purity:
0.98
SMILES:
Cl.C[C@@H]1CCCN1CCCOc1ccc(cc1)-c1ccc(=O)[nH]n1