TargetMol

EGFR-IN-52

Product Code:
 
TAR-T61646
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61646-5mg5mg£1,167.00
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Quantity:
TAR-T61646-50mg50mg£2,307.00
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Quantity:
TAR-T61646-100mg100mg£2,898.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EGFR-IN-52 (Compound 4) is a highly effective inhibitor of the epidermal growth factor receptor (EGFR). It exhibits IC50 values of 0.358, 86.02, and 432.67 uM against EGFR, EGFR L858R-TK, and EGFR T790M-TK, respectively. Additionally, EGFR-IN-52 demonstrates potent cytotoxic effects on cancer cell lines and triggers apoptosis [1].
CAS:
454436-75-0
Formula:
C19H18N4O3S
Molecular Weight:
382.44
Purity:
0.98
SMILES:
Cc1c(NC(=S)Nc2ccc3OCOc3c2)c(=O)n(-c2ccccc2)n1C