TargetMol

MA242 free base

Product Code:
 
TAR-T62977
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T62977-5mg5mg£1,167.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T62977-50mg50mg£2,307.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T62977-100mg100mg£2,898.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
MA242 free base is a specific dual inhibitor of MDM2 and NFAT1 that induces apoptosis in pancreatic cancer cell lines. MA242 free base binds directly to MDM2 and NFAT1 with high affinity, induces MDM2 and NFAT1 protein degradation and inhibits NFAT1-mediated MDM2 transcription.
CAS:
1049704-17-7
Molecular Weight:
465.95
Purity:
0.98
SMILES:
Cc1ccc(cc1)S(=O)(=O)n1cc2CCN=C3C=C(NCc4ccc(Cl)cc4)C(=O)c1c23