TargetMol

Henatinib

Product Code:
 
TAR-T63011
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T63011-5mg5mg£1,167.00
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Quantity:
TAR-T63011-50mg50mg£2,307.00
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Quantity:
TAR-T63011-100mg100mg£2,898.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Henatinib is an orally active small molecule multi-kinase inhibitor with broad antitumour effects. henatinib inhibits the activity of VEGFR-2 (IC50: 0.6 nM), c-kit (IC50: 3.3 nM), PDGFR (IC50: 41.5 nM). henatinib significantly inhibits VEGFR-2 phosphorylation and its downstream signalling pathways in human umbilical vein endothelial cells (HUVECs). Henatinib significantly inhibited VEGFR-2 phosphorylation and its downstream signaling pathway in human umbilical vein endothelial cells (HUVECs).
CAS:
1239269-51-2
Molecular Weight:
468.529
Purity:
0.98
SMILES:
Cc1c(\C=C2/C(=O)Nc3ccc(F)cc23)[nH]c2CCCN(C[C@H](O)CN3CCOCC3)C(=O)c12