TargetMol

MS8511

Product Code:
 
TAR-T63351
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T63351-5mg5mg£850.00
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Quantity:
TAR-T63351-50mg50mg£1,661.00
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Quantity:
TAR-T63351-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
MS8511 is a selective G9a/GLP covalent irreversible inhibitor by targeting a cysteine residue at the substrate binding site, with IC 50 values of 100 nM (G9a) and 140 nM (GLP), and K d values of 44 nM (G9a) and 46 nM (GLP). MS8511 reduces the cellular H3K9me2 level and enhances antiproliferation activity. MS8511 can be used for the research of several types of cancers including brain, breast, ovarian, lung, bladder, melanoma, colorectal cancer , and other disease such as Alzheimer?s disease (AD), sickle cell disease, Prader-Willi syndrome (PWS) [1] .
CAS:
2866408-21-9
Molecular Weight:
495.66
Purity:
0.98