TargetMol

dBRD4-BD1

Product Code:
 
TAR-T69506
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T69506-5mg5mg£1,171.00
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TAR-T69506-50mg50mg£2,303.00
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Quantity:
TAR-T69506-100mg100mg£3,042.00
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Further Information

Bioactivity:
dBRD4-BD1 is a selective BRD4 bromodomain inhibitor. dBRD4-BD1 can selectively degrade BRD4 (DC50 = 280 nM). Notably, dBRD4-BD1 upregulates BRD2/3, a result not observed with degraders using pan-BET ligands. Designing BRD4 selectivity up front enables analysis of BRD4 biology without wider BET-inhibition and simplifies designing BRD4-selective heterobifunctional molecules, such as degraders with new E3 recruiting ligands or for additional probes beyond degraders.
CAS:
2839318-19-1
Molecular Weight:
967.02
Purity:
0.98