TargetMol

Glucocorticoid receptor modulator 1

Product Code:
 
TAR-T72102
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T72102-5mg5mg£284.00
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Quantity:
TAR-T72102-50mg50mg£1,155.00
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Quantity:
TAR-T72102-100mg100mg£1,797.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Glucocorticoid receptor modulator 1 is a highly potent and orally active non-steroidal selective glucocorticoid receptor modulator with an IC 50 value of 9 nM and 130 nM for NF-κB and AP-1 , respectively. Glucocorticoid receptor modulator 1 can effectively reduce the expression of inflammatory factors IL-6 , IL-1β, TNF-α, also can relieve dermatitis in mice .
CAS:
2868357-11-1
Molecular Weight:
470.97
Purity:
0.98
SMILES:
O=C(C=1C=CC=CC1)N2C3=CC=C(C=C3CCC2)NS(=O)(=O)C=4C=C(Cl)C(=CC4OC)C