TargetMol

EGFR-IN-61

Product Code:
 
TAR-T73128
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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CodeSizePrice
TAR-T73128-5mg5mg£850.00
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Quantity:
TAR-T73128-50mg50mg£1,661.00
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Quantity:
TAR-T73128-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EGFR-IN-61 is a potent EGFR kinase inhibitor, with IC 50 values of 42 nM (L858R/T790 M), 137 nM (L858R/T790 M/C797S), and 743 nM (WT), respectively. EGFR-IN-61 shows antiproliferative activity against A549 and H1975 cell lines, with IC 50 values of 2.14 and 1.82 uM, respectively .
Molecular Weight:
629.15
Purity:
0.98
SMILES:
CN(C)CCN(C)C1=CC(=C(C=C1NC(=O)C2=CC(=NC=C2)Cl)NC3=NC=CC(=N3)C4=CN(C5=CC=CC=C54)CCCO)OC