TargetMol

PROTAC BRD4 Degrader-17

Product Code:
 
TAR-T74270
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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TAR-T74270-50mg50mgEnquire
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TAR-T74270-5mg5mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PROTAC BRD4 Degrader-17 (compound 13i) is a potent PROTAC BRD4 Degrader, with IC 50 values of 29.54 nM ( BRD4 (BD1) ) and 3.82 nM ( BRD4 (BD2) ). PROTAC BRD4 Degrader-17 significantly attenuates G2/M progression associated Cyclin B1 expression. PROTAC BRD4 Degrader-17 significantly induces apoptosis in MV-4-11 cells [1] .
CAS:
2585561-49-3
Molecular Weight:
877.94
Purity:
0.98