TargetMol

USP28-IN-2

Product Code:
 
TAR-T74792
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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CodeSizePrice
TAR-T74792-50mg50mgEnquire
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TAR-T74792-5mg5mgEnquire
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
USP28-IN-2 is a USP28 inhibitor ( IC 50 =0.3 uM) with high selectivity over USP2, USP7, USP8 , USP9x, UCHL3 and UCHL5. USP28-IN-2 shows cytotoxicity against cancer cells, down-regulates the cellular level of c-Myc through ubiquitin-proteasome system. USP28-IN-2 also decreases the ankyrase-1/2 level in vitro . USP28-IN-2 enhance the sensitivity of colorectal cancer cells to Regorafenib [1] .
Molecular Weight:
475.39
Purity:
0.98