TargetMol

Pactimibe sulfate

Product Code:
 
TAR-T62974
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T62974-25mg25mg£1,163.00
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Quantity:
TAR-T62974-50mg50mg£1,765.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Pactimibe sulfate (CS-505) is a dual ACAT1/2 inhibitor, acting on ACAT1 (IC50: 4.9 uM) and ACAT2 (IC50: 3.0 uM). Pactimibe sulfate inhibited oleoyl-CoA non-competitively (Ki: 5.6 uM) and significantly inhibited cholesterol ester formation (IC50: 6.7 uM). Pactimibe sulfate reduces plasma cholesterol activity and has anti-atherogenic potential.
CAS:
608510-47-0
Molecular Weight:
931.28
Purity:
0.98
SMILES:
OS(O)(=O)=O.CCCCCCCCN1CCc2c1c(NC(=O)C(C)(C)C)c(C)c(CC(O)=O)c2C.CCCCCCCCN1CCc2c1c(NC(=O)C(C)(C)C)c(C)c(CC(O)=O)c2C