TargetMol

KG-548

Product Code:
 
TAR-T60539
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T60539-100mg100mgEnquire
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TAR-T60539-50mg50mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
KG-548 is an ARNT/TACC3 disruptor as well as a HIF-1α inhibitor. KG-548 directly interferes with the formation of the ARNT/TACC3 complex by competitively binding the ARNT PAS-B domain with TACC3. ARNT is the aryl hydrocarbon receptor nuclear translocator which is also known as HIF-β [1][2].
CAS:
175205-09-1
Molecular Weight:
282.149
Purity:
0.98
SMILES:
FC(F)(F)C1=CC(=CC(=C1)C(F)(F)F)C2=NN=NN2