TargetMol

PF-06761281

Product Code:
 
TAR-T60547
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T60547-100mg100mgEnquire
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T60547-50mg50mgEnquire
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • Show All

Further Information

Bioactivity:
PF-06761281 (Compound 4a) is a potent, orally active, partial selective inhibitor of sodium-coupled citrate transporter (NaCT or SLC13A5). The IC50 values of HEK NaCT, HEK NaDC1, and HEK NaDC3 are 0.51, 13.2 and 14.1 uM, respectively [1].
CAS:
1854061-19-0
Molecular Weight:
283.28
Purity:
0.98
SMILES:
COc1ncc(C)cc1CC[C@@](O)(CC(O)=O)C(O)=O