TargetMol

GPR81 agonist 1

Product Code:
 
TAR-T62656
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T62656-50mg50mg£1,364.00
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Quantity:
TAR-T62656-100mg100mg£1,990.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GPR81 agonist 1 is a highly selective and potent GPR81 agonist that acts in human (IC50: 58 nM) and mouse (IC50: 50 nM). GPR81 agonist 1 is more selective for GPR81 than GPR109a. GPR81 agonist 1 inhibits lipolysis in mice and does not cause skin flushing.
CAS:
1620992-67-7
Molecular Weight:
446.63
Purity:
0.98
SMILES:
C[C@H]1CC[C@@H](CC1)C(=O)Nc1nc(c(CC(=O)N2CCN(C)CC2)s1)-c1cccs1