TargetMol

APS-2-79

Product Code:
 
TAR-T70004
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T70004-100mg100mgEnquire
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TAR-T70004-50mg50mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
APS-2-79 is a KSR -dependent MEK antagonist. APS-2-79 inhibits ATP biotin binding to KSR2 within the KSR2-MEK1 complexe with an IC 50 of 120 nM. APS-2-79 makes the stabilization of the KSR inactive state antagonizes oncogenic Ras-MAPK signaling .
CAS:
2002381-25-9
Molecular Weight:
387.43
Purity:
0.98
SMILES:
N=1C=NC(NC2=CC=C(OC=3C=CC=CC3)C=C2C)=C4C=C(OC)C(OC)=CC14