TargetMol

BAY-3827

Product Code:
 
TAR-T73350
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T73350-100mg100mgEnquire
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TAR-T73350-50mg50mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
BAY-3827 is a potent and selective AMPK inhibitor with IC 50 values of 1.4 nM at low (10 uM ATP concentration) and 15 nM at high (2 mM ATP concentration). BAY-3827 shows over 500-fold selectivity for most of the 331 kinases. BAY-3827 prevents phosphorylation of acetyl-CoA carboxylase 1 and shows strongest anti-proliferative activity in androgen-dependent prostate cancer cell lines .
CAS:
2377576-35-5
Molecular Weight:
468.53
Purity:
0.98
SMILES:
N#CC1=C(N(C(=C(C#N)C1C2=CC=3C(=NNC3C(=C2F)C)NC(=O)C=4C=CC=CC4CC)C)C)C