TargetMol

Sitagliptin phosphate monohydrate

Product Code:
 
TAR-T0242L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T0242L-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T0242L-100mg100mg£111.00
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Further Information

Bioactivity:
Sitagliptin phosphate is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.
CAS:
654671-77-9
Formula:
C16H15F6N5O?H3PO4?H2O
Molecular Weight:
523.32
Pathway:
Proteases/Proteasome|Autophagy|Ubiquitination
Purity:
0.9965
SMILES:
C1CN2C(=NN=C2C(F)(F)F)CN1C(=O)C[C@@H](CC3=CC(=C(C=C3F)F)F)N.O.OP(=O)(O)O
Target:
DPP-4|Autophagy|Proteasome

References

Kim SJ et al. Diabetes. 2009; 58(3): 641-651. Thomas L et al. J Pharmacol Exp Ther. 2008; 325(1): 175-182.