TargetMol

PROTAC ER Degrader-4

Product Code:
 
TAR-T13839
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T13839-100mg100mgEnquire
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TAR-T13839-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).
CAS:
2361114-15-8
Formula:
C53H67F3N6O8S
Molecular Weight:
1005.2
Purity:
0.98
SMILES:
C(C(C)(C)F)N1[C@@](C2=C(C=3C(N2)=CC=CC3)C[C@H]1C)(C4=C(F)C=C(OCCOCCOCCOCC(N[C@H](C(=O)N5[C@H](C(N[C@@H](C)C6=CC=C(C=C6)C7=C(C)N=CS7)=O)C[C@@H](O)C5)C(C)(C)C)=O)C=C4F)[H]

References

Bin Yang, et al. Compounds and their use in treating cancer. WO2019123367A1.