TargetMol

Ketanserinol

Product Code:
 
TAR-T25568
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T25568-100mg100mgEnquire
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TAR-T25568-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
Ketanserinol is the metabolite of ketanserin. Ketanserin is a hypotensive drug with 5-HT2 receptor antagonism, used to reverse pulmonary hypertension caused by protamine.
CAS:
76330-73-9
Molecular Weight:
397.44
Purity:
0.98
SMILES:
O=C1NC=2C=CC=CC2C(=O)N1CCN3CCC(CC3)C(O)C4=CC=C(F)C=C4

References

Yassen A, Hanff LM, Vulto AG. Simultaneous quantitative analysis of ketanserin and ketanserinol in plasma by RP-HPLC with fluorescence detection. Biomed Chromatogr. 2003 Dec;17(8):517-21. PubMed PMID: 14648608. Frenken M, Kaumann AJ. Interaction of ketanserin and its metabolite ketanserinol with 5HT2 receptors in pulmonary and coronary arteries of calf. Naunyn Schmiedebergs Arch Pharmacol. 1984 Jul;326(4):334-9. PubMed PMID: 6482982. Schoenwald RD, Zhu J. The ocular pharmacokinetics of ketanserin and its metabolite, ketanserinol, in albino rabbits. J Ocul Pharmacol Ther. 2000 Oct;16(5):481-95. PubMed PMID: 11110040. Kurowski M. Simultaneous determination of ketanserin and ketanserinol in biological fluids using ion-pair liquid chromatography and fluorometric detection. J Chromatogr. 1985 May 31;341(1):208-12. PubMed PMID: 3160719.