Metkephamid

Product Code:

TAR-T25804

Product Group:

Inhibitors and Activators

Supplier:

TargetMol

Regulatory Status:

RUO

Shipping:

cool pack

Storage:

-20°C

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Code	Size	Price

TAR-T25804-100mg

100mg

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TAR-T25804-500mg

500mg

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Further Information

Bioactivity:

Metkephamid is a synthetic opioid pentapeptide and derivative of [Met]enkephalin. It shows as a potent agonist of the δ- and u-opioid receptors with roughly equipotent affinity, and also has similarly high affinity as well as subtype-selectivity for the κ3-opioid receptor.

CAS:

66960-34-7

Molecular Weight:

600.73

Purity:

0.98

SMILES:

[C@H](CC1=CC=CC=C1)(C(N([C@@H](CCSC)C(N)=O)C)=O)NC(CNC([C@H](NC([C@H](CC2=CC=C(O)C=C2)N)=O)C)=O)=O

Documents

References

Leander JD, Wood CR. Metkephamid effects on operant behavior. Peptides. 1982 Sep-Oct;3(5):771-3. PubMed PMID: 7177922. Bloomfield SS, Barden TP, Mitchell J. Metkephamid and meperidine analgesia after episiotomy. Clin Pharmacol Ther. 1983 Aug;34(2):240-7. PubMed PMID: 6872419. Pasanisi F, Sloan L, Rubin PC. Cardiovascular properties of metkephamid, a delta opioid receptor agonist, in man. Clin Sci (Lond). 1985 Feb;68(2):209-13. PubMed PMID: 2981652. Burkhardt C, Frederickson RC, Pasternak GW. Metkephamid (Tyr-D-ala-Gly-Phe-N(Me)Met-NH2), a potent opioid peptide: receptor binding and analgesic properties. Peptides. 1982 Sep-Oct;3(5):869-71. PubMed PMID: 6294639.