TargetMol

PSB-1011 sodium

Product Code:
 
TAR-T28461
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T28461-100mg100mgEnquire
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TAR-T28461-500mg500mgEnquire
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Further Information

Bioactivity:
PSB-1011 is a selective and competitive inhibitor of the rat P2X2 receptor (Ki = 79 nM).
CAS:
08/01/4499
Molecular Weight:
683.4
Purity:
0.98
SMILES:
[Na].[Na].Nc1c(cc(Nc2ccc(c(Nc3nc(Cl)nc(Cl)n3)c2)S(O)(=O)=O)c2C(=O)c3ccccc3C(=O)c12)S(O)(=O)=O

References

Baqi Y, Hausmann R, Rosefort C, Rettinger J, Schmalzing G, M?ller CE. Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem. 2011 Feb 10;54(3):817-30. Epub 2011 Jan 5. PubMed PMID: 21207957. Hausmann R, Schmalzing G. P2X1 and P2X2 receptors in the central nervous system as possible drug targets. CNS Neurol Disord Drug Targets. 2012 Sep;11(6):675-86. Review. PubMed PMID: 22963438.