TargetMol

S-MGB-234 TFA

Product Code:
 
TAR-T34663
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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This product comes from: United States.
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Further Information

Bioactivity:
S-MGB-234 is a novel Minor Groove Binder that cures animal African trypanosomiasis in an in vivo mouse model. S-MGB-234 has significant potential as novel therapeutic agents for animal African trypanosomiasis.
CAS:
1970223-54-1
Molecular Weight:
796.67
Purity:
0.98
SMILES:
OC(C(F)(F)F)=O.O=C(C1=CC(NC(C2=CN=C(/C=C/C3=CC=C(C=C3)OC)C=C2)=O)=CN1C)NC4=CN(C)C(C(NCCC(N)=N)=O)=C4.OC(C(F)(F)F)=O

References

Giordani F, Khalaf AI, Gillingwater K, Munday JC, de Koning HP, Suckling CJ, Barrett MP, Scott FJ. Novel Minor Groove Binders cure animal African trypanosomiasis in an in vivo mouse model. J Med Chem. 2019 Feb 14. doi: 10.1021/acs.jmedchem.8b01847. [Epub ahead of print] PubMed PMID: 30763102.