TargetMol

BRD4 ligand-Linker Conjugate 1

Product Code:
 
TAR-T39629
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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Further Information

Bioactivity:
BRD4 Ligand-Linker Conjugate 1 is a compound consisting of a ligand and a linker, specifically designed to bind to the target protein BRD4. This conjugate serves as a valuable tool for synthesizing PROTACs, molecules utilized for targeted protein degradation.
CAS:
2154358-89-9
Molecular Weight:
500.05
Purity:
0.98
SMILES:
Cc1nnc2n1-c1ccc(cc1C(=NC21CC1)c1ccc(Cl)cc1)-c1cnn(CCCCCCN)c1 |c:14|

References

Sun D, et al. Evaluation of the Small-molecule BRD4 Degrader CFT-2718 in Small-cell Lung Cancer and Pancreatic Cancer Models. Mol Cancer Ther. 2021 Aug;20(8):1367-1377.