TargetMol

PROTAC CDK9 degrader-4

Product Code:
 
TAR-T39996
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T39996-100mg100mgEnquire
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TAR-T39996-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
PROTAC CDK9 degrader-4 is a potent and efficacious chemical compound designed specifically to degrade CDK9, a protein involved in transcription regulation. This compound effectively targets and reduces the levels of CDK9, thereby modulating transcriptional activity.
CAS:
2411021-01-5
Molecular Weight:
792.986
Purity:
0.98
SMILES:
CC[C@@H](CO)Nc1cc(NCc2ccc(NC(=O)N3CCN(CCCCCc4cccc5C(=O)N(Cc45)C4CCC(=O)NC4=O)CC3)cc2)n2ncc(C(C)C)c2n1

References

Wei D, et al. Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer. J Med Chem. 2021 Oct 14;64(19):14822-14847.