TargetMol

Pralsetinib HCl (2097132-94-8 free base)

Product Code:
 
TAR-TQ0277L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-TQ0277L-100mg100mgEnquire
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TAR-TQ0277L-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
Pralsetinib is a selective and next-generation RET inhibitor (IC50: 0.3-0.4 nM for WT RET, RET mutants V804L, V804M, M918T, and CCDC6-RET fusion). BLU-667 is an effective and selective inhibitor of RET mutations, fusions, and predicted resistant mutants.
CAS:
TQ0277L
Molecular Weight:
570.07
Purity:
0.98
SMILES:
O=C([C@@]1(OC)CC[C@@H](C2=NC(NC3=NNC(C)=C3)=CC(C)=N2)CC1)N[C@H](C4=CC=C(N5N=CC(F)=C5)N=C4)C.[H]Cl