AdipoGen Life Sciences

PIK-90

Product Code:
 
SYN-1068
Product Group:
 
Inhibitors and Activators
Regulatory Status:
 
RUO
Shipping:
 
-20°C
1 / 1
Chemical Structure
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Chemical Structure

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SYN-1068-M100100 mgEnquire
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SYN-1068-M0011 mg£69.00
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SYN-1068-M0055 mg£92.00
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SYN-1068-M01010 mg£151.00
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SYN-1068-M05050 mg£426.00
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Further Information

Alternate Names/Synonyms:
PIK90
Appearance:
Solid.
CAS:
677338-12-4
EClass:
32160000
Form (Short):
liquid
InChi:
InChI=1S/C18H17N5O3/c1-25-13-6-5-12-14(15(13)26-2)21-18(23-9-8-20-16(12)23)22-17(24)11-4-3-7-19-10-11/h3-7,10H,8-9H2,1-2H3,(H,21,22,24)
InChiKey:
ZJAVHOMVDCMAMF-UHFFFAOYSA-N
Long Description:
Chemical. CAS: 677338-12-4. Formula: C18H17N5O3. MW: 351.4. PIK-90 is a potent PI3K inhibitor with IC(50) values of 11, 18, and 58nM for p110alpha, gamma and delta isoforms respectively. It has an IC(50) of 350nM for the p110beta isoform. It also has low mTOR activity.
Molecular Formula:
C18H17N5O3
Molecular Weight:
351.4
Package Type:
Plastic Vial
Product Description:
PIK-90 is a potent PI3K inhibitor with IC(50) values of 11, 18, and 58nM for p110alpha, gamma and delta isoforms respectively. It has an IC(50) of 350nM for the p110beta isoform. It also has low mTOR activity.
Purity:
>95%
Solubility Chemicals:
Slightly soluble (<1mg/ml) in DMSO or ethanol.
Transportation:
Non-hazardous
UNSPSC Category:
Protein Kinase Modulators
UNSPSC Number:
12352200
Use & Stability:
Stable for at least 2 years after receipt when stored at -20°C.

References

A pharmacological map of the PI3-K family defines a role for p110alpha in insulin signaling: Z.A. Knight, et al.; Cell 125, 733 (2006)