TargetMol

AS2717638

Product Code:
 
TAR-T10381
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10381-1mg1mg£189.00
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TAR-T10381-5mg5mg£329.00
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TAR-T10381-1mL1 mL * 10 mM (in DMSO)£354.00
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TAR-T10381-10mg10mg£503.00
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TAR-T10381-25mg25mg£768.00
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TAR-T10381-50mg50mg£1,018.00
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Quantity:
TAR-T10381-100mg100mg£1,348.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5). It also significantly improves PGF2α-, PGE2-, and AMPA-induced allodynia.
CAS:
2148339-28-8
Formula:
C25H25N3O5
Molecular Weight:
447.48
Purity:
0.9867
SMILES:
O=C1C=2C=C(OC)C(OC)=CC2C(=CN1C3=NOC=4C=CC(=CC43)C)C(=O)N5CCCCC5

References

1. Murai N, et al. Analgesic effects of novel lysophosphatidic acid receptor 5 antagonist AS2717638 in rodents. Neuropharmacology. 2017 Nov;126:97-107.