EMPA

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TargetMol
Product Code: TAR-T11186
Supplier: TargetMol
CodeSizePrice
TAR-T11186-1mg1mg£108.00
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TAR-T11186-5mg5mg£168.00
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TAR-T11186-1mL1 mL * 10 mM (in DMSO)£177.00
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TAR-T11186-10mg10mg£229.00
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TAR-T11186-25mg25mg£436.00
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TAR-T11186-50mg50mg£610.00
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TAR-T11186-100mg100mg£838.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM respectively)
CAS:
680590-49-2
Formula:
C23H26N4O4S
Molecular Weight:
454.55
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9991
SMILES:
CCN(Cc1cccnc1)C(=O)CN(c1ccc(OC)nc1)S(=O)(=O)c1ccccc1C
Target:
OX Receptor

References

1. P Malherbe, et al. Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX