NF-56-EJ40

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TargetMol
Product Code: TAR-T12216
Supplier: TargetMol
CodeSizePrice
TAR-T12216-1mg1mg£137.00
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TAR-T12216-5mg5mg£229.00
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TAR-T12216-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T12216-10mg10mg£334.00
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TAR-T12216-25mg25mg£519.00
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TAR-T12216-50mg50mg£703.00
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TAR-T12216-100mg100mg£970.00
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TAR-T12216-500mg500mg£1,862.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.
CAS:
2380230-73-7
Formula:
C27H29N3O3
Molecular Weight:
443.547
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.98
SMILES:
CN1CCN(Cc2ccc(cc2)-c2cccc(c2)C(=O)Nc2ccccc2CC(O)=O)CC1
Target:
GPR

References

1. Haffke M, et al. Structural basis of species-selective antagonist binding to the succinate receptor. Nature. 2019 Oct;574(7779):581-585.