TK216

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TargetMol
Product Code: TAR-T13166
Supplier: TargetMol
CodeSizePrice
TAR-T13166-1mg1mg£100.00
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TAR-T13166-5mg5mg£142.00
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TAR-T13166-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T13166-10mg10mg£195.00
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TAR-T13166-25mg25mg£322.00
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TAR-T13166-50mg50mg£503.00
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TAR-T13166-100mg100mg£695.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.
CAS:
1903783-48-1
Formula:
C19H15Cl2NO3
Molecular Weight:
376.23
Pathway:
; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Purity:
0.9845
SMILES:
OC1(CC(=O)c2ccc(cc2)C2CC2)C(=O)Nc2c1c(Cl)ccc2Cl
Target:
DNA/RNA Synthesis

References

1. Spriano F, et al. The ETS Inhibitors YK-4-279 and TK-216 Are Novel Antilymphoma Agents. Clin Cancer Res. 2019 Aug 15;25(16):5167-5176. 2. Brian Lannutti, et al. Uses of indolinone compounds. US10159660B2.