BI-3812

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TargetMol
Product Code: TAR-T14561
Supplier: TargetMol
CodeSizePrice
TAR-T14561-1mg1mg£173.00
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TAR-T14561-2mg2mg£217.00
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TAR-T14561-5mg5mg£282.00
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TAR-T14561-1mL1 mL * 10 mM (in DMSO)£330.00
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TAR-T14561-10mg10mg£430.00
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TAR-T14561-25mg25mg£664.00
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TAR-T14561-50mg50mg£863.00
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TAR-T14561-100mg100mg£1,187.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
BI-3812 is an inhibitor of BCL6. Which inhibiting the BTB domain of BCL6 (IC50: 3 nM). BI-3812 also has antitumor activity.
CAS:
2166387-64-8
Formula:
C26H32ClN7O5
Molecular Weight:
558.04
Pathway:
Apoptosis
Purity:
0.9979
SMILES:
CNC(=O)COc1cc2cc(Nc3nc(ncc3Cl)N3CCC(CC3)C(=O)N(C)C)cc(OC)c2n(C)c1=O
Target:
BCL

References

1. Kerres N, et al. Chemically Induced Degradation of the Oncogenic Transcription Factor BCL6. Cell Rep. 2017 Sep 19;20(12):2860-2875.