DBPR108

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TargetMol
Product Code: TAR-T15079
Supplier: TargetMol
CodeSizePrice
TAR-T15079-1mg1mg£166.00
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TAR-T15079-5mg5mg£309.00
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TAR-T15079-1mL1 mL * 10 mM (in DMSO)£333.00
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TAR-T15079-10mg10mg£389.00
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TAR-T15079-25mg25mg£603.00
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TAR-T15079-50mg50mg£830.00
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TAR-T15079-100mg100mg£1,099.00
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TAR-T15079-500mg500mg£2,135.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.
CAS:
1186426-66-3
Formula:
C16H25FN4O2
Molecular Weight:
324.4
Pathway:
Ubiquitination; Proteases/Proteasome
Purity:
0.9965
SMILES:
CC(C)(CC(=O)N1CCCC1)NCC(=O)N1C[C@@H](F)C[C@H]1C#N
Target:
Proteasome; DPP-4

References

1. Yeh TK, et al. (2S,4S)-1-[2-(1,1-dimethyl-3-oxo-3-pyrrolidin-1-yl-propylamino)acetyl]-4-fluoro-pyrrolidine-2-carbonitrile: a potent, selective, and orally bioavailable dipeptide-derived inhibitor of dipeptidyl peptidase IV. Bioorg Med Chem Lett. 2010 Jun