Delgocitinib

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TargetMol
Product Code: TAR-T15096
Supplier: TargetMol
CodeSizePrice
TAR-T15096-1mg1mg£209.00
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Quantity:
TAR-T15096-1mL1 mL * 10 mM (in DMSO)£365.00
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Quantity:
TAR-T15096-5mg5mg£503.00
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Quantity:
TAR-T15096-10mg10mg£695.00
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Quantity:
TAR-T15096-25mg25mg£1,018.00
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Quantity:
TAR-T15096-50mg50mg£1,348.00
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Quantity:
TAR-T15096-100mg100mg£1,813.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Delgocitinib is a novel and specific inhibitor of JAK (IC50s: 2.8, 2.6, 13 and 58 nM for JAK1, JAK2, JAK3 and Tyk2, respectively) .
CAS:
1263774-59-9
Formula:
C16H18N6O
Molecular Weight:
310.361
Pathway:
Tyrosine Kinase/Adaptors; JAK/STAT signaling; Angiogenesis; Stem Cells; Chromatin/Epigenetic
Purity:
0.999
SMILES:
C[C@H]1CN(C(=O)CC#N)[C@]11CCN(C1)c1ncnc2[nH]ccc12
Target:
Tyrosine Kinases; JAK

References

1. Tanimoto A, et al. Pharmacological properties of JTE-052: a novel potent JAK inhibitor that suppresses various inflammatory responses in vitro and in vivo. Inflamm Res. 2015 Jan;64(1):41-5