Mutant IDH1 inhibitor

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TargetMol
Product Code: TAR-T16161
Supplier: TargetMol
CodeSizePrice
TAR-T16161-1mg1mg£125.00
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TAR-T16161-5mg5mg£205.00
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TAR-T16161-1mL1 mL * 10 mM (in DMSO)£219.00
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TAR-T16161-10mg10mg£302.00
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TAR-T16161-25mg25mg£460.00
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TAR-T16161-50mg50mg£627.00
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TAR-T16161-100mg100mg£863.00
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TAR-T16161-500mg500mg£1,653.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
CAS:
1429180-08-4
Formula:
C25H34N6O3
Molecular Weight:
466.586
Pathway:
Metabolism
Purity:
0.9772
SMILES:
CC(C)[C@H]1COC(=O)N1c1ccnc(N[C@@H](C)c2ccc(CN3CCN(CC3)C(C)=O)cc2)n1
Target:
Dehydrogenase; Isocitrate Dehydrogenase (IDH)

References

1. 3-Pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH and their preparation. Patent WO 2013046136 A1 20130404