Vidupiprant

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TargetMol
Product Code: TAR-T17232
Supplier: TargetMol
CodeSizePrice
TAR-T17232-1mg1mg£119.00
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TAR-T17232-5mg5mg£189.00
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TAR-T17232-1mL1 mL * 10 mM (in DMSO)£230.00
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TAR-T17232-10mg10mg£254.00
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TAR-T17232-25mg25mg£405.00
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TAR-T17232-50mg50mg£570.00
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TAR-T17232-100mg100mg£781.00
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TAR-T17232-500mg500mg£1,500.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Vidupiprant is an effective dual antagonist of CRTH2 and prostanoid D receptor with IC50s of 8 nM and 35 nM in human plasma. Vidupiprant can be used in studies about the treatment of asthma.
CAS:
1169483-24-2
Formula:
C28H27Cl2FN2O6S
Molecular Weight:
609.49
Pathway:
GPCR/G Protein; Immunology/Inflammation
Purity:
0.98
SMILES:
CC(C)(C)NC(=O)c1ccc(Oc2cc(F)c(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(cc2Cl)C2CC2)c1
Target:
Prostaglandin Receptor

References

1. Liu J, et al. Discovery of AMG 853, a CRTH2 and DP Dual Antagonist. ACS Med Chem Lett. 2011 Mar 2;2(5):326-30.