ELN-441958

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TargetMol
Product Code: TAR-T2086
Supplier: TargetMol
CodeSizePrice
TAR-T2086-1mg1mg£145.00
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TAR-T2086-2mg2mg£181.00
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TAR-T2086-5mg5mg£254.00
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TAR-T2086-1mL1 mL * 10 mM (in DMSO)£274.00
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TAR-T2086-10mg10mg£369.00
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TAR-T2086-25mg25mg£576.00
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TAR-T2086-50mg50mg£790.00
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TAR-T2086-100mg100mg£1,050.00
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TAR-T2086-500mg500mg£2,038.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958 is highly selective for B1 over B2 receptors.
CAS:
913064-47-8
Formula:
C29H29ClN4O2
Molecular Weight:
501.03
Pathway:
GPCR/G Protein
Purity:
0.989
SMILES:
Clc1cccc2CN(C(=O)c12)c1cccc(c1)C(=O)N1CCC2(CC1)CCN(CC2)c1ccncc1
Target:
Bradykinin Receptor

References

1. Hawkinson JE, et al. J Pharmacol Exp Ther.2007 Aug;322(2):619-630.