APD668

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TargetMol
Product Code: TAR-T2088
Supplier: TargetMol
CodeSizePrice
TAR-T2088-1mg1mg£111.00
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TAR-T2088-2mg2mg£130.00
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TAR-T2088-5mg5mg£168.00
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TAR-T2088-1mL1 mL * 10 mM (in DMSO)£174.00
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TAR-T2088-10mg10mg£230.00
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TAR-T2088-25mg25mg£374.00
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TAR-T2088-50mg50mg£518.00
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TAR-T2088-100mg100mg£691.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.
CAS:
832714-46-2
Formula:
C21H24FN5O5S
Molecular Weight:
477.51
Pathway:
GPCR/G Protein; Endocrinology/Hormones; Membrane transporter/Ion channel; Metabolism
Purity:
0.9997
SMILES:
CC(C)OC(=O)N1CCC(CC1)Oc1ncnc2n(ncc12)-c1ccc(cc1F)S(C)(=O)=O
Target:
GPR; P45; Potassium Channel

References

1. Semple G, et al. Bioorg Med Chem Lett. 2011 May 15;21(10):3134-41.