MK-1064

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TargetMol
Product Code: TAR-T3722
Supplier: TargetMol
CodeSizePrice
TAR-T3722-1mg1mg£122.00
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TAR-T3722-5mg5mg£195.00
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TAR-T3722-1mL1 mL * 10 mM (in DMSO)£214.00
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TAR-T3722-10mg10mg£275.00
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TAR-T3722-25mg25mg£477.00
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TAR-T3722-50mg50mg£646.00
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TAR-T3722-100mg100mg£846.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
MK-1064 is a selective orexin 2 receptor antagonist (2-SORA).
CAS:
1207253-08-4
Formula:
C24H20ClN5O3
Molecular Weight:
461.91
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9988
SMILES:
COc1ccc(CNC(=O)c2cc(cnc2-c2ccccn2)-c2cncc(Cl)c2)nc1OC
Target:
OX Receptor

References

Roecker AJ et al. ChemMedChem. 2014 Feb;9(2):311-22. Gotter AL et al. Orexin 2 Receptor Antagonism is Sufficient to Promote NREM and REM Sleep from Mouse to Man. Sci Rep. 2016 Jun 3;6:27147.