Obafistat

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TargetMol
Product Code: TAR-T39635
Supplier: TargetMol
CodeSizePrice
TAR-T39635-1mg1mg£124.00
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TAR-T39635-5mg5mg£201.00
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TAR-T39635-1mL1 mL * 10 mM (in DMSO)£213.00
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TAR-T39635-10mg10mg£282.00
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TAR-T39635-25mg25mg£470.00
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TAR-T39635-50mg50mg£651.00
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TAR-T39635-100mg100mg£863.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4).
CAS:
2160582-57-8
Formula:
C15H16FN5O3S
Molecular Weight:
365.38
Pathway:
Metabolism
Purity:
0.98
SMILES:
O=C(c1cnn[nH]1)N(CC1CC2)CC2N1S(c1cc(F)ccc1)(=O)=O
Target:
NADPH

References

Marcus Koppitz, et al. [8-(phenylsulfonyl)-3,8-diazabicyclo[3.2.1]oct-3-yl] (1h-1,2,3-triazol-4-yl)methanones. WO2017202817A1.